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Linagliptin-d4
Cat. No. IC23100
CAS. No. 2140263-92-7
Key Features and Details
Category
Inhibitor&Activator
Formula
C25H24D4N8O2
Product Details
Product Name
Linagliptin-d4
CAS No.
2140263-92-7
Molecular Weight
476.57
Synonyms
BI 1356-d4
Formula
C25H24D4N8O2
SMILES
CC#CCN1C2=C(N(C(N(C2=O)CC3=NC4=C(C=CC=C4)C(C)=N3)=O)C)N=C1N5C([2H])([2H])[C@@H](CCC5([2H])[2H])N
Product Overview
Description
Linagliptin-d4 is deuterium labeled Linagliptin. Linagliptin is a highly potent, selective DPP-4 inhibitor with IC50 of 1 nM.
In Vitro Activity
Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.
Storage & Handling
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Shipping
Room temperature in continental US; may vary elsewhere.
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