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Linagliptin-13C,d3
Cat. No. IC23096
CAS. No. 1398044-43-3
Key Features and Details
Category
Inhibitor&Activator
Formula
C2413CH25D3N8O2
Product Details
Product Name
Linagliptin-13C,d3
CAS No.
1398044-43-3
Molecular Weight
476.55
Synonyms
BI 1356-13C,d3
Formula
C2413CH25D3N8O2
SMILES
[2H][13C]([2H])([2H])C#CCN1C2=C(N(C(N(C2=O)CC3=NC4=C(C=CC=C4)C(C)=N3)=O)C)N=C1N5C[C@@H](CCC5)N
Product Overview
Description
Linagliptin-13C,d3 is the 13C- and deuterium labeled Linagliptin. Linagliptin is a highly potent, selective DPP-4 inhibitor with IC50 of 1 nM.
In Vitro Activity
Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.
Storage & Handling
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Shipping
Room temperature in continental US; may vary elsewhere.
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