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TCS PIM-1 4a (SMI-4a)
Product Name: | TCS PIM-1 4a (SMI-4a) |
CAT#: | DEP-2312-LGZ-3 |
Package: | 10mg/25mg/50mg/10mM * 1mL in DMSO |
Datasheet |
Description
TCS Pim-1 4a is a selective and ATP-competitive Pim kinase inhibitor with IC50 values of 24 and 100 nM for Pim-1 and Pim-2, respectively.
Basic Information
Application: | Pim Inhibitor |
CAS Number: | 438190-29-5 |
Formula: | C11H6F3NO2S |
Molecular Weight: | 273.23 |
SMILES: | O=C(NC/1=O)SC1=C\C2=CC=CC(C(F)(F)F)=C2 |
Solubility-In vitro: | In vitro (25°C): DMSO: 47 mg/mL (172.01 mM) Water: Insoluble Ethanol: 28 mg/mL (102.47 mM) |
Solubility-In vivo: | 30% PEG400+0.5% Tween80+5% propylene glycol: 28 mg/mL |
Target Info
Pim1: | 17 nM |
Storage
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Preparing Stock Solutions
0.1 mM_1 mg: 36.6 mL
0.1 mM_5 mg: 183 mL
0.1 mM_10 mg: 365.99 mL
0.5 mM_1 mg: 7.32 mL
0.5 mM_5 mg: 36.6 mL
0.5 mM_10 mg: 73.2 mL
1 mM_1 mg: 3.66 mL
1 mM_5 mg: 18.3 mL
1 mM_10 mg: 36.6 mL
5 mM_1 mg: 0.73 mL
5 mM_5 mg: 3.66 mL
5 mM_10 mg: 7.32 mL
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