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TCS PIM-1 4a (SMI-4a)

Product Name: TCS PIM-1 4a (SMI-4a)
CAT#: DEP-2312-LGZ-3
Package: 10mg/25mg/50mg/10mM * 1mL in DMSO


TCS Pim-1 4a is a selective and ATP-competitive Pim kinase inhibitor with IC50 values of 24 and 100 nM for Pim-1 and Pim-2, respectively.

Basic Information

Application: Pim Inhibitor
CAS Number: 438190-29-5
Formula: C11H6F3NO2S
Molecular Weight: 273.23
Solubility-In vitro: In vitro (25°C):
DMSO: 47 mg/mL (172.01 mM)
Water: Insoluble
Ethanol: 28 mg/mL (102.47 mM)
Solubility-In vivo: 30% PEG400+0.5% Tween80+5% propylene glycol: 28 mg/mL

Target Info

Pim1: 17 nM


  • The lyophilized form should be stored at -20°C, in a desiccated environment.
  • In lyophilized form, the chemical remains stable for 36 months.
  • In solution, it should be stored at -20°C and used within 3 months to prevent loss of potency. Aliquoting is recommended to avoid multiple freeze/thaw cycles.

Preparing Stock Solutions

0.1 mM_1 mg: 36.6 mL 0.1 mM_5 mg: 183 mL 0.1 mM_10 mg: 365.99 mL 0.5 mM_1 mg: 7.32 mL 0.5 mM_5 mg: 36.6 mL 0.5 mM_10 mg: 73.2 mL 1 mM_1 mg: 3.66 mL 1 mM_5 mg: 18.3 mL 1 mM_10 mg: 36.6 mL 5 mM_1 mg: 0.73 mL 5 mM_5 mg: 3.66 mL 5 mM_10 mg: 7.32 mL

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