Histone Acetyltransferase Inhibitor II

Product Name:	Histone Acetyltransferase Inhibitor II
CAT#:	DEHA-2312-LGZ-1
Package:	5mg/10mg/50mg/100mg
Datasheet

Description

Histone acetyltransferase inhibitor II is a highly effective cell-permeable p300 inhibitor with an IC50 of 5 μM, and can be used in cancer research.

Basic Information

Application:	p300 Inhibitor
CAS Number:	932749-62-7
Formula:	C20H16Br2O3
Molecular Weight:	464.15
SMILES:	O=C1/C(CCC/C1=C\C2=CC=C(O)C(Br)=C2)=C/C3=CC=C(O)C(Br)=C3
*Solubility-In vitro:*	DMSO: 82 mg/mL (176.66 mM) Water: Insoluble Ethanol: 18 mg/mL * <1 mg/ml means slightly soluble or insoluble.

Storage

The lyophilized form should be stored at -20°C, in a desiccated environment.
In lyophilized form, the chemical remains stable for 36 months.
In solution, it should be stored at -20°C and used within 3 months to prevent loss of potency. Aliquoting is recommended to avoid multiple freeze/thaw cycles.

Preparing Stock Solutions

0.1 mM_1 mg: 21.54 mL 0.1 mM_5 mg: 107.72 mL 0.1 mM_10 mg: 215.45 mL 0.5 mM_1 mg: 4.31 mL 0.5 mM_5 mg: 21.54 mL 0.5 mM_10 mg: 43.09 mL 1 mM_1 mg: 2.15 mL 1 mM_5 mg: 10.77 mL 1 mM_10 mg: 21.54 mL 5 mM_1 mg: 0.43 mL 5 mM_5 mg: 2.15 mL 5 mM_10 mg: 4.31 mL

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.